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Drug DiscoveryStructure-Activity RelationshipAmerican Chemical SocietyMedicinal ChemistryPeptides and ProteinsBiological EvaluationOrally BioavailableDrug DesignMetabolic StabilityLead OptimizationKinase InhibitorsLead CompoundKinase Inhibitorin Vitro and in VivoNovel SeriesSmall-molecule InhibitorsPharmacokinetic PropertiesVirtual ScreeningRay CrystallographyInhibitory Activity
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